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Glycin-Plasmamembran-Transportproteine
Eintrag öffnenGlyxambi · 4.5 · An interaction study with gemfibrozil, an in vitro inhibitor of OAT3 and OATP1B1/1B3 transporters, showed that
Eintrag öffnenGlyxambi · 4.5 · Inhibition of OATP1B1/1B3 transporters by co-administration with rifampicin resulted in a 75% increase in Cmax
Eintrag öffnenHepcludex · 4.5 · In vitro an inhibition of OATP1B1/3 transporters by bulevirtide was observed, albeit only at a concentration ≥
Eintrag öffnenIbrance · 4.5 · In vitro studies with transporters
Eintrag öffnenIbrance · 4.5 · In vitro studies with transporters
Eintrag öffnenInrebic · 4.5 · Effects on transporters In in vitro studies, fedratinib inhibits P-glycoprotein (P-gp), breast cancer resistan
Eintrag öffnenJakavi · 4.5 · Substances transported by P-glycoprotein or other transporters Ruxolitinib may inhibit P-glycoprotein and brea
Eintrag öffnenJakavi · 4.5 · Substances transported by P-glycoprotein or other transporters Ruxolitinib may inhibit P-glycoprotein and brea
Eintrag öffnenJardiance · 4.5 · An interaction study with gemfibrozil, an in vitro inhibitor of OAT3 and OATP1B1/1B3 transporters, showed that
Eintrag öffnenJardiance · 4.5 · Empagliflozin does not inhibit human uptake transporters such as OAT3, OATP1B1, and OATP1B3 in vitro at clinic
Eintrag öffnenJardiance · 4.5 · Inhibition of OATP1B1/1B3 transporters by co-administration with rifampicin resulted in a 75% increase in Cmax
Eintrag öffnenJentadueto · 4.5 · 7 Organic cation transporters (OCT) Metformin is a substrate of both transporters OCT1 and OCT2. Co-administra
Eintrag öffnenJoenja · 4.5 · BCRP inhibitors Leniolisib is a substrate of BCRP transporters. No interaction studies have been conducted wit
Eintrag öffnenJuluca · 4.5 · In vitro, dolutegravir inhibited the renal uptake transporters, organic anion transporters (OAT)1 and OAT3. Ba
Eintrag öffnenJyseleca · 4.5 · Filgotinib is not a clinically relevant inhibitor or inducer of most enzymes or transporters commonly involved
Eintrag öffnenK Cl- Cotransporters
Eintrag öffnenKaftrio · 4.5 · 9 In vitro studies showed that TEZ is a substrate for the uptake transporter OATP1B1 and efflux transporters P
Eintrag öffnenKaftrio · 4.5 · In vitro studies showed that TEZ is a substrate for the uptake transporter OATP1B1 and efflux transporters P-g
Eintrag öffnenKaftrio · 4.5 · Potential for interaction with transporters Co-administration of IVA or TEZ/IVA with digoxin, a sensitive P-gp
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