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Atazanavir Viatris (previously Atazanavir Mylan) · 4.5 · Atazanavir is an inhibitor of CYP3A4. The potential inhibition of P-gp by atazanavir is unknown and cannot be
Eintrag öffnenAtazanavir Viatris (previously Atazanavir Mylan) · 4.5 · Atazanavir is metabolised in the liver through CYP3A4. It inhibits CYP3A4. Therefore, atazanavir is contraindi
Eintrag öffnenAtazanavir Viatris (previously Atazanavir Mylan) · 4.5 · Lomitapide Lomitapide is highly dependent on CYP3A4 Co-administration of for metabolism and co-administration
Eintrag öffnenAtazanavir Viatris (previously Atazanavir Mylan) · 4.5 · The mechanism of diltiazem/atazanavir interaction is CYP3A4 inhibition. Verapamil Serum concentrations of vera
Eintrag öffnenAtazanavir Viatris (previously Atazanavir Mylan) · 4.5 · The mechanism of interaction between atazanavir and ritonavir is CYP3A4 inhibition. Indinavir Indinavir is ass
Eintrag öffnenAtazanavir Viatris (previously Atazanavir Mylan) · 4.5 · The mechanism of the clarithromycin/atazanavir interaction is CYP3A4 inhibition. ANTIFUNGALS Ketoconazole 200
Eintrag öffnenAtectura Breezhaler · 4.5 · Inhibition of CYP3A4 and P-glycoprotein (P-gp) has no impact on the safety of therapeutic doses of Atectura Br
Eintrag öffnenAtectura Breezhaler · 4.5 · Inhibition of the key contributors of indacaterol clearance (CYP3A4 and P-gp) or mometasone furoate clearance
Eintrag öffnenAtectura Breezhaler · 4.5 · Interaction with CYP3A4 and P-glycoprotein inhibitors
Eintrag öffnenAugtyro · 4.5 · Based on in vitro data repotrectinib is a substrate for CYP3A4 and P-gp.
Eintrag öffnenAugtyro · 4.5 · Effect of CYP3A4 and P-gp inducers on repotrectinib Co-administration of multiple oral doses of rifampicin (a
Eintrag öffnenAugtyro · 4.5 · Effect of CYP3A4 inhibitors and P-gp inhibitors on repotrectinib Co-administration of multiple oral doses of i
Eintrag öffnenAugtyro · 4.5 · Effect of repotrectinib on CYP3A4 substrates Repotrectinib is a moderate CYP3A4 inducer. Co-administration of
Eintrag öffnenAugtyro · 4.5 · Oral contraceptives Repotrectinib is a moderate CYP3A4 inducer, which can decrease progestin or oestrogen expo
Eintrag öffnenAvamys · 4.5 · Based on data with another glucocorticoid (fluticasone propionate), that is metabolised by CYP3A4, coadministr
Eintrag öffnenAzarga · 4.5 · The cytochrome P-450 isozymes responsible for metabolism of brinzolamide include CYP3A4 (main), CYP2A6, CYP2B6
Eintrag öffnenAzopt · 4.5 · 4 The cytochrome P-450 isozymes responsible for metabolism of brinzolamide include CYP3A4 (main), CYP2A6, CYP2
Eintrag öffnenBalversa · 4.5 · Grapefruit or Seville oranges should be avoided while taking Balversa due to strong CYP3A4 inhibition (see sec
Eintrag öffnenBalversa · 4.5 · Moderate CYP2C9 or strong CYP3A4 inhibitors Co-administration with a moderate CYP2C9 or strong CYP3A4 inhibito
Eintrag öffnenBalversa · 4.5 · Strong or moderate CYP3A4 inducers Co-administration with carbamazepine, a strong CYP3A4 and weak CYP2C9 induc
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