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Balversa · 4.5 · Organic cation transporter 2 (OCT2) substrates Mean ratios of Cmax and AUC∞ for metformin (a sensitive OCT2 su
Eintrag öffnenBiktarvy · 4.5 · Bictegravir inhibits organic cation transporter 2 (OCT2) and multidrug and toxin extrusion transporter 1 (MATE
Eintrag öffnenCresemba · 4.5 · Isavuconazole is a mild inhibitor of the organic cation transporter 2 (OCT2). Co-administration of isavuconazo
Eintrag öffnenCresemba · 4.5 · Isavuconazole is a mild inhibitor of the organic cation transporter 2 (OCT2). Co-administration of isavuconazo
Eintrag öffnenDovato · 4.5 · In vitro, dolutegravir inhibited the renal transporters OCT2 and MATE1. In vivo, a 10-14% decrease of creatini
Eintrag öffnenDovato · 4.5 · In vitro, lamivudine was an inhibitor of OCT1 and OCT2; the clinical consequences are not known.
Eintrag öffnenDovato · 4.5 · Lamivudine is cleared renally. Active renal secretion of lamivudine in the urine is mediated through the OCT2
Eintrag öffnenErleada · 4.5 · Based on in vitro data, inhibition of organic cation transporter 2 (OCT2), organic anion transporter 3 (OAT3)
Eintrag öffnenErleada · 4.5 · Based on in vitro data, inhibition of organic cation transporter 2 (OCT2), organic anion transporter 3 (OAT3)
Eintrag öffnenFampyra · 4.3 · Concomitant use of Fampyra with medicinal products that are inhibitors of Organic Cation Transporter 2 (OCT2)
Eintrag öffnenHalaven · 4.5 · At relevant clinical concentrations, eribulin did not inhibit BCRP, OCT1, OCT2, OAT1, OAT3, OATP1B1 and OATP1B
Eintrag öffnenJentadueto · 4.5 · 7 Organic cation transporters (OCT) Metformin is a substrate of both transporters OCT1 and OCT2. Co-administra
Eintrag öffnenJuluca · 4.5 · In vitro, dolutegravir inhibited the renal organic cation transporter 2 (OCT2) and multidrug and toxin extrusi
Eintrag öffnenLynparza · 4.5 · In vitro, olaparib has been shown to be an inhibitor of BCRP, OATP1B1, OCT1, OCT2, OAT3, MATE1 and MATE2K. It
Eintrag öffnenMaviret · 4.5 · Significant inhibition of CYP1A2, CYP2C9, CYP2C19, CYP2D6, UGT1A6, UGT1A9, UGT1A4, UGT2B7, OCT1, OCT2, OAT1, O
Eintrag öffnenMaviret · 4.5 · Significant inhibition of CYP1A2, CYP2C9, CYP2C19, CYP2D6, UGT1A6, UGT1A9, UGT1A4, UGT2B7, OCT1, OCT2, OAT1, O
Eintrag öffnenMethylthioninium chloride Proveblue · 4.5 · Methylthioninium chloride is a potent inhibitor of the transporters OCT2, MATE1 and MATE2-K. The clinical cons
Eintrag öffnenMysimba · 4.5 · Bupropion and its metabolites competitively inhibit the OCT2 in the basolateral membrane of the renal tubule r
Eintrag öffnenMysimba · 4.5 · OCT2 substrates
Eintrag öffnenOrganischer Kationen-Transporter 2
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